Browsing by Author "Cabedo, Nuria"
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Andreu, Inmaculada; Cortes, Diego; Protais, Philippe; Cassels Niven, Bruce; Chagraoui, Abdeslam; Cabedo, Nuria (Elsevier Science Ltd., 1999-11-15)AbstractÐThe preparation of N-methyl-BTHIQ (4) from N-phenylethyl-phenacetamide (1) by cyclization, reduction and N-alkyl- ation in acid medium has been achieved in good yield in a `one-pot' procedure. Acylation of imine ...
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Cabedo, Nuria; Protais, Philippe; Cassels Niven, Bruce; Cortes, Diego (American Chemical Society and American Society of Pharmacognosy, 1998-01-15)(R)-(+)-nor-Roefractine (1) was synthesized by the Bischler-Napieralski route, using asymmetric reduction of the 1,2-didehydro precursor imine with sodium (S)-N-CBZ-prolinyloxyborohydride. Compound 1 was able to displace ...